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Pharm II
MOA/Receptors
41
Pharmacology
Graduate
09/12/2014
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Term
Amantadine
 Definition
Enhances exiting Dopa
NMDA Antagonist
Cholinergic Receptor Antagonist
Parksinsons
Term
Levodopa and Carvidopa
 Definition
Pre-dopamine substrate
Dopa Mimetic
Parkinsons
Term
Selegilline
 Definition
Inhibits MAO-B
Parksinons
Term
Rasagilline (azilect)
 Definition
Inhibits MAO-B
Parksinsons
Term
Tolcapone (Tasmar)
 Definition
Inhibits COMT
Parksinsons
Term
Entacapone (Comtan)
 Definition
Inhibits COMT
Parkinsons
Term
Bromocriptine(pariodel)
 Definition
D1 and D2 agonist (ergot)
Parkinsons
Term
Pramipexole (mirapex)
 Definition
D2 agonist
Parkinsons
Term
Ropinirole (requip)
 Definition
D2 agonist
Parkinsons
Term
Rotigotine (neupro)
 Definition
D2 agonist
Parkinsons
Term
Apomorphine (apokyn)
 Definition
D- agonist for off-eposides
Dopamine Agonist
Parkinsons
Term
Benztropine(cogentin)
 Definition
Block excitatory M-receptors, restore balance with Dopamine
Anti-Muscurcinic
Parkinsons
Term
Biperiden (artane)
 Definition
Block excitatory M-receptors, restore balance with Dopamine
Antimuscurinic
Parkinsons
Term
Akineton (trihexyphenydyl)
 Definition
Block excitatory M-receptors, restore balance with Dopamine
Anti-Muscurinic
Parkinsons
Term
Donepezil (aricept)
 Definition
Inhibit AChE, somewhat specially in CNS
Alzheimers
Term
Galantamine
 Definition
Inhibit AChE, somewhat specially in CNS
Alzheimers
Term
Rivastigmine
 Definition
Inhibit AChE, somewhat specially in CNS
Alzheimers
Term
Tacrine
 Definition
Inhibit AChE, somewhat specially in CNS
Alzheimers
Term
Glutamate
 Definition
Inhibit NMDA Receptors
Alzheimers
Term
Memantine (namenda)
 Definition
Inhibit NMDA receptors
Alzheimers
Term
Oxazepam (serax)
 Definition
Inhibitory effect on GABA receptors via allosteric site
Benzodiazepines- anti-anxiety
SA
Term
Triazolamn (halcoin)
 Definition
Inhibitory effect on GABA receptors via allosteric site
Benzodiazepines- anti-anxiety
SA
Term
Midazolam (versed)
 Definition
Inhibitory effect on GABA receptors via allosteric site
Benzodiazepines- anti-anxiety
SA
Term
Alprazolam (xanax)
 Definition
Inhibitory effect on GABA receptors via allosteric site
Benzodiazepines- anti-anxiety
IA
Term
Temazepam (restoril)
 Definition
Inhibitory effect on GABA receptors via allosteric site
Benzodiazepines- anti-anxiety
IA
Term
Lorazepam (ativan)
 Definition
Inhibitory effect on GABA receptors via allosteric site
Benzodiazepines- anti-anxiety
IA
Term
Diazepam (valium)
 Definition
Inhibitory effect on GABA receptors via allosteric site
Benzodiazepines- anti-anxiety
LA
Term
Flurazepam (dalmane)
 Definition
Inhibitory effect on GABA receptors via allosteric site
Benzodiazepines- anti-anxiety
LA
Term
Clonazepam (Klonopin)
 Definition
Inhibitory effect on GABA receptors via allosteric site
Benzodiazepines- anti-anxiety
LA
Term
Chlordiazepoxide (librium)
 Definition
Inhibitory effect on GABA receptors via allosteric site
Benzodiazepines- anti-anxiety
LA
Term
Clorazepate(Tranxene)
 Definition
Inhibitory effect on GABA receptors via allosteric site
Benzodiazepines- anti-anxiety
LA
Term
Flumazenil
 Definition
BZ antagonist
BZ overdose agent
Term
Zolpidem (ambien)
 Definition
Subset of BZ site of GABA receptors
Sedatives
anxiolytic / hypnotic
Term
Lunesta
 Definition
Subset of BZ site of GABA receptors
Sedatives
Anxiolytic/hypnotic
Term
Ramelton (Rozerem)
 Definition
Melatonin MT1 and MT2 agonist
Sedative
Anxiolytic/ hypnotic
Term
Hydroxyzine
 Definition
Antihistamine (H1 first generation)
sedative
anxiolytic hypnotic
Term
Buspirone (BusPar)
 Definition
5HT 1A/2A and D2 agonist
GAD
anxiolytic/hypnotic
Term
thiopental
 Definition
GABA hyperpolirzation via non - BZ receptor
Barbituates
Term
Penobarbital
 Definition
GABA hyperpolerization via non- BZ receptor
barbituate
Term
Chloral Hydrate
 Definition
???
Non Barbituate
Term
Disulfiram
 Definition
Block aldehyde
Non-Barb
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