Term
Acetylcholine (Miochol-E)
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Definition
Direct Acting Muscarinic Agonist
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Term
Carbachol (Isopto Carbachol)
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Definition
Direct Acting Muscarinic Agonist
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Term
Methacholine (Provocholine)
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Definition
Direct Acting Muscarinic Agonist
- pulmonary function testing in asthma
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Term
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Definition
Direct Acting Muscarinic Agonist
- GI motility
- Treat urine retention
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Term
pilocarpine (Salagen/Ocusert Pilo)
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Definition
Direct Acting Muscarinic Agonist
- Treat glaucoma
- Treat xerostomia
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Term
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Definition
Reversible cholinesterase inhibitor
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Term
physostigmine/eserine (Antilirium)
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Definition
Reversible cholinesterase inhibitor
- Antidote to antimuscarinic OD
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Term
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Definition
Reversible cholinesterase inhibitor
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Term
pyridostigmine (Mestinon)
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Definition
Reversible cholinesterase inhibitor
- Treat MG
- Pre-exposure protection by army
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Term
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Definition
Reversible cholinesterase inhibitor
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Term
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Definition
Reversible cholinesterase inhibitor
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Term
| carbamate insecticides (Carbaryl) |
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Definition
reversible cholinesterase inhibitor |
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Term
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Definition
Irreversible cholinesterase inhibitors
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Term
| Organophosphate insecticides (Parathion, Malathion) |
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Definition
| Irreversible cholinesterase inhibitors |
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Term
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Definition
| Irreversible cholinesterase inhibitors |
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Term
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Definition
| cGMP phosphodiesterase inhibitors |
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Term
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Definition
| cGMP phosphodiesterase inhibitors |
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Term
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Definition
| cGMP phosphodiesterase inhibitors |
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Term
Pralidoxime/2-p AM (Protopam)
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Definition
Cholinesterase Reactivator
- Counters organophosphates (given within 2 hours)
- Counters nerve agents like Sarin
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Term
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Definition
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Term
Atropine, Hyoscyamine and Homatropine
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Definition
Muscarinic antagonists (Anticholinergics)
- Antidote to ACH OD
- Preoperative to block vagal to heart
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Term
| scopolamine and methscopolamine |
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Definition
Muscarinic antagonists (Anticholinergics)
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Term
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Definition
Muscarinic antagonists (Anticholinergics)
- Intestinal antispasmatic for IBS
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Term
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Definition
Muscarinic antagonists (Anticholinergics)
- GI antispasmdic to treat IBS
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Term
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Definition
Muscarinic antagonists (Anticholinergics)
- anesthetic to dry secretions
- inhibit vagal reflexes
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Term
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Definition
Muscarinic antagonists (Anticholinergics)
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Term
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Definition
Muscarinic antagonists (Anticholinergics)
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Term
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Definition
Muscarinic antagonists (Anticholinergics)
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Term
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Definition
Muscarinic antagonists (Anticholinergics)
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Term
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Definition
Muscarinic antagonists (Anticholinergics)
- Treat urinary incontinence
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Term
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Definition
Muscarinic antagonists (Anticholinergics)
- Treat urinary incontinence
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Term
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Definition
Muscarinic antagonists (Anticholinergics)
- Treat urinary incontinence
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Term
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Definition
Muscarinic antagonists (Anticholinergics)
- DIalate pupil for eye exams
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Term
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Definition
Competative (nondepolarizing blocker)
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Term
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Definition
Selective β1-agonist
- Treat cardiogenic shock
- Start heart back up again
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Term
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Definition
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Term
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Definition
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Term
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Definition
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Term
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Definition
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Term
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Definition
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Term
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Definition
Selective α1-agonists
- Dilate eyes without causing cycloplagia
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Term
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Definition
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Term
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Definition
| Indirect-acting Sympathomimetics |
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Term
| Pseudoephedrine (Sudafed) |
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Definition
Indirect-acting Sympathomimetics
- Treat stress induced urinary incontinance
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Term
A woman takes a med to lower her BP, which worsens her reynaud's symptoms. Which drug caused this?
- Reserpine
- Metoprolol
- Methyldopa
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Definition
- Reserpine
- Metoprolol
- Methyldopa
Reynaud's is worsened by peripheral β1 blockers.
Reserpine is a peripheral neuronal blocker.
Methyldopa is a central neuronal blocker.
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Term
Which drug will block both alpha and beta?
- Labetalol
- Esmolol
- Atenolol
- Metoprolol
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Definition
- Labetalol (α,β)
- Esmolol (β1)
- Atenolol (β1)
- Metoprolol (β1)
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Term
A drug that selectively stimulates B1 and is used to start the heart back up is
- Albuterol
- Phenylepherine
- Dobutamine
- Terbutaline
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Definition
- Albuterol (β2)
- Phenylepherine (α1)
- Dobutamine (β1)
- Terbutaline (β2)
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Term
Clonidine cures all EXEPT
- Hypertension
- Migraine
- Morphine withdrawal
- Urinary incontinence
- spinal analgesic-like effect
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Definition
- Hypertension
- Migraine
- Morphine withdrawel
- Urinary incontinance
- spinal analgesic-like effect
Also for ADHD, hot flahes, PTSD
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Term
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Definition
- Prazosin
- Terazosin
- Doxazosin
- Tamsulosin
- Alfuzosin
- Silodosin
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Term
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Definition
- Prazosin
- Terazosin
- Doxazosin
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Term
| Treat Urinary incontinence |
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Definition
- Solifenacin (Vesicare)
- Pseudoephedrine
- Oxybutynin
- Tolterodine
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Term
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Definition
- Propantheline
- Dicyclomine (Bentyl)
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Term
| Prevent hypertension during Pheochromocytoma |
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Definition
- Phenoxybenzamine
- Phentolamine
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Term
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Definition
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Term
|
Definition
- Pramipexole (Mirapex)
- Ropinerole (Requip)
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Term
|
Definition
- Nadolol
- Phenoxybenzamine
- Reserpine
- Cialis
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Term
|
Definition
- Trihexyphenidyl (Artane)
- Benztropine (Cogentin)
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Term
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Definition
- Detect: Edrophonum (Tensilon)
- Neostigmine
- Pyridostigmine
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Term
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Definition
- Donepezil (Aricept)
- Rivastigmine (Exelon)
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Term
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Definition
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Term
| Lowers BP by stimulating A2 receptors in brain |
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Definition
- Clonidine
- Guanfacine
- Methyldopa
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Term
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Definition
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Term
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Definition
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Term
| Which drug is used to relax the uterus and prevent premature labor? |
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Definition
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Term
| A drug that can be used as a local anesthetic with vasoconstrictor properties because of it's indirect sympathomametic activity is |
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Definition
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Term
A patient is given a drug for his hypertension that may cause orthostatic hypotension on the first day
the drug is |
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Definition
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Term
| drug used to counter tissue necrosis |
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Definition
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Term
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Definition
- Selegiline (Eldepryl)
- Deprenyl (Zelapar)
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Term
| which drug is used to distinguish between myesthenia crisis and cholinergic crisis? |
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Definition
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Term
| Stopage of this has no rebound since it acts on NT stored in vessicles (LA) |
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Definition
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Term
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Definition
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Term
| Drug which decreases lactation |
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Definition
Bromocriptine (parlodel)
second choice for parkinsen's |
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Term
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Definition
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Term
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Definition
B2 agonist
+ Terbutaline
+ Metaproterenol |
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Term
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Definition
Direct acting muscarinic agonist
+ Pilocarpine |
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Term
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Definition
Reversible cholinesterase inhibitor
+ Aricept
+ Carbamate insectacides (Carbaryl) |
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Term
| Antidote to antimuscarinic OD |
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Definition
| Physostigmine (Antilirium) |
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Term
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Definition
| Methacholine (Provocholine) |
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Term
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Definition
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Term
Acebutolol (Sectral)
- Blocks
- Partial agonist?
- Membrane stabalizing?
- Lipid solubility?
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Definition
- β1 blocker
- partial agonist
- membrane stabilizing
- Low lipid solubility
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Term
Atenolol (Tenormin)
- Blocks
- Partial agonist?
- Membrane stabalizing?
- Lipid solubility?
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Definition
- β1 blocker
- Not partial agonist
- Not membrane stabalizing
- Low lipid solubility
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Term
Esmolol (Brevibloc)
- Blocks
- Partial agonist?
- Membrane stabalizing?
- Lipid solubility?
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Definition
- Blocks β1
- Not partial agonist
- Not membrane stabalizing
- Low lipid solubility
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Term
Metoprolol (Lopressor, Toprol XL)
- Blocks
- Partial agonist?
- Membrane stabalizing?
- Lipid solubility?
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Definition
- Blocks β1
- Not partial agonist
- Membrane stabalizing
- Medium Lipid solubility
Worsens raynaulds
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Term
Nadolol (Corgard)
- Blocks
- Partial agonist?
- Membrane stabalizing?
- Lipid solubility?
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Definition
- Blocks β1 & β2
- Not Partial agonist
- Non Membrane stabalizing
- Low lipid solubility
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Term
Pindolol
- Blocks
- Partial agonist?
- Membrane stabalizing?
- Lipid solubility?
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Definition
- Blocks β1, β2
- Partial agonist
- Membrane stabalizing
- Medium lipid solubility?
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Term
Propranolol (Inderal-LA)
- Blocks
- Partial agonist?
- Membrane stabalizing?
- Lipid solubility?
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Definition
- Blocks β1, β2
- not Partial agonist
- Membrane stabalizing
- High lipid solubility
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Term
Timolol (Timoptic)
- Blocks
- Partial agonist?
- Membrane stabalizing?
- Lipid solubility?
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Definition
- Blocks β1,β2
- Not partial agonist
- Not membrane stabalizing
- Medium lipid solubility
- Treat glaucoma
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Term
|
Definition
- Blocks α, β
- Treat hypertension
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Term
Phenoxybenzamine (Dibenzyline)
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Definition
- Non selective α1,α2 blocker
- Non competative LA inhibitor
- prevent hypertension during pheochromocytoma
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Term
|
Definition
- Non selective α1α2 blocker
- Treat pheochromocytoma
- Counter tissue necrosis
- counter oral anesthetics
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Term
|
Definition
- Selective α1 blocker
- Treat hypertension
- Treat BPH
- Treat raynauds
- treat PTSD
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Term
|
Definition
- Selective α1 blocker
- Treat hypertension
- Treat BPH
- Treat raynauds
- treat PTSD
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Term
|
Definition
- Selective α1 blocker
- Treat hypertension
- Treat BPH
- Treat raynauds
- treat PTSD
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Term
|
Definition
- Selective α1 blocker
- Treat BPH
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Term
|
Definition
- Selective α1 blocker
- Treat BPH. Acumulate in prostate
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Term
|
Definition
- Selective α1 blocker
- Treat BPH
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Term
|
Definition
- peripheral acting sympathetic neuronal blocker
- Decrease NE, Da into vessicles. LA
- Lowers BP
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Term
|
Definition
- Centrally acting sympathetic neuronal blocker
- prodrug. α agonist at CNS to lowr outflow of sympatheti activity
- lower renin release
- treat hypertension during pregnancy
- induce autoimmune disorders
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Term
|
Definition
- Centrally acting sympathetic neuronal blocker
- patch
- lowers BP, migraine, ADHD, PTSD, hot flashes
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Term
| Guanfacine (Tenex, Intuniv) |
|
Definition
- Centrally acting sympathetic neuronal blocker
- less rebound than clonidine
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Term
Nicotine
- Heart
- Vessels
- Eye
- GI
- Bladder
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Definition
(Ganglionic stimulant)
- Heart: Tachycardia, ↓ contractility
- Vessels: vasodilation, ↓TPR
- Eye: Mydriasis, cycloplegia
- GI: ↓tone, motility, secretion
- Bladder: urine retention
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|
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Term
|
Definition
|
|
Term
| l-dopa + Carbidopa (Sinemet) |
|
Definition
|
|
Term
l-dopa + Carbidopa +Entacapone
(Stalevo) |
|
Definition
|
|
Term
|
Definition
- Dopaminergic agent
- second choice, less on-off
- decreases lactation
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Term
|
Definition
- Dopaminergic agent
- Also usefull for restless leg
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Term
|
Definition
- Dopaminergic agent
- also usefull for RLS
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Term
|
Definition
- Dopaminergic agent
- Stimulate release of dopamine.
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Term
| Selegiline/Deprenyl (Eldepryl, Zelapar) |
|
Definition
|
|
Term
|
Definition
|
|
Term
| Diphenhydramine (benadryl) |
|
Definition
- Antihistamine
- blocks muscarinic as SE
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