| Term 
 | Definition 
 
        | Muscarinic agonist, orally -selective for M3 in GI and bladder
 *stimulate intestine and bladder
 *ex. urinary retention (will promote micturition)
 Contraindicated:
 -asthmatic
 -peptic ulcers
 -coronary insufficiency
 |  | 
        |  | 
        
        | Term 
 | Definition 
 
        | Muscarinic agonist -1st choice for open angle glaucoma
 |  | 
        |  | 
        
        | Term 
 
        | Carbachol (Carbamylcholine) |  | Definition 
 
        | Muscarinic agonist -open angle glaucoma
 SE: impaired night vision (contracts ciliary muscles of the eye for near vision, miosis)
 |  | 
        |  | 
        
        | Term 
 | Definition 
 
        | nonselective Muscarinic Antagonist *use: cholinesterase poisoning (life saving short term because it blocks muscarinic effects)
 -crosses BBB poorly
 
 in general
 -overactive bladder
 -anti-parinsonian treatment
 |  | 
        |  | 
        
        | Term 
 | Definition 
 
        | Muscarinic Antagonist -methylated atropine
 *Use: anesthetic adjuvant, motion sickness
 -potent muscarinic antagonist with INCREASED CNS activity
 |  | 
        |  | 
        
        | Term 
 | Definition 
 
        | Muscarinic Antagonist -spec. for M1 subtype--> ULCERS
 |  | 
        |  | 
        
        | Term 
 | Definition 
 
        | Muscarinic Antagonist -bronchodilation
 |  | 
        |  | 
        
        | Term 
 | Definition 
 
        | Muscarinic Antagonist -bronchodilation
 |  | 
        |  |