Term
| BZD used for anxiety that has a cyclopropyl group |
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Definition
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Term
| BZD used primarily for anxiety that has a trifluromethyl group |
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Definition
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Term
| BZD used for insomnia that has a tertiary amine group |
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Definition
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Term
| BZD Prodrug of oxazepam used for PARTIAL seizures, anxiety and withdrawal symptoms that has a carboxyl group at C-3 |
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Definition
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Term
| Thioamide (-N-C=O-C=S-)BZD that contains a trifluromethyl group used primarily for insomnia that has a trifluromethyl group |
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Definition
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Term
| BZD used to treat all types of seizure EXCEPT grand mal that contains a nitro group |
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Definition
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Term
| BZD that can undergo hydrolysis into a lactam N----->O |
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Definition
| Chlordiazepoxide (Librax, Librium) |
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Term
| BZDs containing a triazole ring that is used for many types of seizures EXCEPT grand mal |
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Definition
| Triazolam, Alprazolam, Estazolam |
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Term
| BZD containing an imidazole ring used for preoperative sedation and for IV anesthesia |
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Definition
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Term
| NonBZD carbamate sleep aid that has a chiral center and only the S configuration is used. |
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Definition
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Term
| Non-BZD sleep aid with shorten sleep latency, prolonged sleep time and has no effect on stages of sleep that contains an imidazopyridine ring |
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Definition
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Term
| BZD competitive antagonist that contains an imidazole ring that is used for BZD overdose (blocks both agonists and inverse agonists) |
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Definition
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Term
| Partial inverse agonist that freezes BZD receptors, close CL- channels and decrease conductance |
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Definition
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Term
| Only Structural difference between Romazicon and RO 15-4513` |
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Definition
| Romazicon has a X=F- and RO 15-4513 has X=N3 |
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Term
| Why is RO 15-4513 considered an agonist and not an antagonist? |
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Definition
| Because it actually binds to a receptor and not just blocks it although it result in antagonistic effects such as closing of CL- channel |
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Term
| Location of serotonin receptors |
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Definition
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